A cell-permeable Ca2? antagonist and vasodilator. Inhibits protein kinase A (Ki = 1.6 μM), protein kinase G (Ki = 1.6 μM), myosin light chain kinase (Ki = 36 μM) and Rho kinase (ROCK; IC50 = 10.7 μM. Fasudil also mobilizes ***** neural stem cells in vivo.
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